SAPHRIS(R) (asenapine) Meets Primary Endpoint in Long-Term Extension Study in Patients With Predominant, Persistent Negative Sym
24 Julio 2009 - 9:07AM
PR Newswire (US)
KENILWORTH, N.J., July 24 /PRNewswire-FirstCall/ -- Schering-Plough
Corporation (NYSE:SGP) today announced that its investigational
agent SAPHRIS(R) (asenapine) met the primary endpoint over one year
of treatment in an extension study in patients with predominant,
persistent negative symptoms of schizophrenia. Negative symptoms of
schizophrenia include apathy, lack of emotion and poor social
functioning, among others. In the study, these symptoms were
assessed using the validated 16-item Negative Symptom Assessment
scale (NSA-16). "These symptoms are among the most difficult to
treat in the schizophrenia spectrum," said Armin Szegedi, M.D.,
Ph.D., vice president, global clinical research, central nervous
system, Schering-Plough Research Institute. "Few studies with the
antipsychotics currently available on the market have been designed
specifically to evaluate long-term effects on predominant,
persistent negative symptoms. The results from this large clinical
study program will provide new insights into potential treatment of
these symptoms." In the study, SAPHRIS was significantly more
effective than olanzapine in the reduction of negative symptoms as
measured by change from baseline to Day 365 in the NSA-16 total
score, the primary endpoint of the study. By using a mixed model
for repeated measures (MMRM), least square mean changes in the
NSA-16 total score were -15.8 for SAPHRIS vs. -11.0 for olanzapine
(P=0.015). Full results of the trial, including efficacy, safety
and tolerability data, will be submitted for presentation at a
medical meeting at a later date. These results follow those of a
previously reported clinical trial in this patient population using
the same study design and protocol in which both asenapine and
olanzapine reduced negative symptoms after one year of treatment,
but the difference between the two was not statistically
significant.(1) Additionally, a preliminary pooled analysis of the
combined data for these two identically designed studies showed a
statistically significant treatment effect in favor of asenapine
after one year of treatment. These large Phase III studies were
conducted following a previous Phase II study where favorable data
on negative symptoms were observed for asenapine. About the study
This study was a 26-week extension of a randomized, double-blind,
multicentered, multinational 26-week clinical trial evaluating the
efficacy and safety of SAPHRIS compared to olanzapine in the
treatment of patients with stable predominant, persistent negative
symptoms of schizophrenia. Patients were initially randomized in
the core study to SAPHRIS 5 to 10 mg twice daily or olanzapine 5 to
20 mg once daily for 26 weeks. In the core study, both SAPHRIS and
olanzapine reduced negative symptoms over the 26-week treatment
period, but the difference between the two was not statistically
significant. Patients who continued after six months were
maintained on the same double-blind treatment regimen for the
26-week extension study. In the extension study, SAPHRIS
demonstrated statistically significantly greater change in NSA-16
total score from the core study baseline after one year of
treatment, the primary prespecified endpoint of the extension
study. A total of 468 patients were randomized in the core study,
195 of whom entered the extension study, with 146 completing a
total of one year of treatment. In the study, the most common
adverse events reported for the SAPHRIS group (greater than 5
percent) during the one year treatment period were: insomnia,
somnolence, weight increase, anxiety, headache, weight decrease,
akathisia, diarrhea, dizziness, fatigue, nasopharyngitis, blood
insulin increase, irritability, dry mouth and nausea. About SAPHRIS
Schering-Plough acquired SAPHRIS in November 2007 through its
acquisition of Organon BioSciences, which developed the
psychotropic agent. In the United States, a New Drug Application
(NDA) for SAPHRIS sublingual tablets is currently under review by
the U.S. Food and Drug Administration (FDA) and includes data from
a clinical trial program involving more than 3,000 patients in
bipolar mania and schizophrenia trials. In Europe, a Marketing
Authorization Application (MAA) for asenapine, under the brand name
SYCREST(R), is currently under review by the European Medicines
Agency (EMEA). About schizophrenia Schizophrenia is a chronic,
disabling brain disorder characterized by hallucinations, delusions
and disordered thinking (often termed positive symptoms), and
cognitive deficits, as well as negative symptoms such as apathy,
avolition, diminished social drive, poverty of speech or curbing of
interest, which are frequent disabling symptoms. About 24 million
people worldwide (or seven in every 1,000 adults in the population)
have schizophrenia, including more than two million people in the
United States and more than four million people in Europe. About
Schering-Plough Schering-Plough is an innovation-driven,
science-centered global health care company. Through its own
biopharmaceutical research and collaborations with partners,
Schering-Plough creates therapies that help save and improve lives
around the world. The company applies its research-and-development
platform to human prescription, animal health and consumer health
care products. Schering-Plough's vision is to "Earn Trust, Every
Day" with the doctors, patients, customers and other stakeholders
served by its colleagues around the world. The company is based in
Kenilworth, N.J., and its Web site is
http://www.schering-plough.com/. SCHERING-PLOUGH DISCLOSURE NOTICE:
The information in this press release includes certain
"forward-looking statements" within the meaning of the Private
Securities Litigation Reform Act of 1995, including statements
relating to the clinical development of, the commercial plans for
and the potential market for SAPHRIS/SYCREST. Forward-looking
statements relate to expectations or forecasts of future events.
Schering-Plough does not assume the obligation to update any
forward-looking statement. Many factors could cause actual results
to differ materially from Schering-Plough's forward-looking
statements, including uncertainties in the regulatory process,
among other uncertainties. For further details about these and
other factors that may impact the forward-looking statements, see
Schering-Plough's Securities and Exchange Commission filings,
including Part II, Item 1A. "Risk Factors" in the Company's first
quarter 2009 10-Q, filed May 1, 2009. Endnote (1) Cazorla P, Phiri
P, den Hollander W, et al. Long-Term Treatment with Asenapine
versus Olanzapine in Subjects with Predominant, Persistent Negative
Symptoms of Schizophrenia. American College of
Neuropsychopharmacology (ACNP) 47th Annual Meeting; Dec. 7-11,
2008; Scottsdale, AZ; No. 88. DATASOURCE: Schering-Plough
Corporation CONTACT: Media: Robert Consalvo, +1-908-298-7409
office, +1-908-295-0928 mobile, or Investors: Janet Barth,
+1-908-298-7436, or Joe Romanelli, +1-908-298-7436 Web Site:
http://www.schering-plough.com/
Copyright